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MS
unreviewed

Pancreatic lipase/colipase, phospholipase A2, cholesterol esterase (+ bile salts)

1 reactions · 1 pathways

Clinical / pharmacological. Suppressed indirectly by corticosteroids (annexin/lipocortin)

What it does, reaction by reaction

1 reactions

Lipoprotein Metabolism (Exogenous and Endogenous Pathways: chylomicrons, VLDL, LDL, HDL) Lipid Metabolism · Intestine, liver, plasma, capillary endothelium

step 1 Irreversible/directional

Dietary TAG, cholesteryl esters, and phospholipids → emulsified mixed micelles

Converts Triacylglycerol (TAG) Cholesteryl ester Phospholipid into Mixed micelle

Notes

In the intestinal lumen, bile salts emulsify dietary lipids; pancreatic lipase with colipase hydrolyzes TAG predominantly to 2-monoacylglycerol plus fatty acids, phospholipase A2 hydrolyzes phospholipids, and cholesterol esterase hydrolyzes cholesteryl esters. This digestive stage is required for absorption but is not a lipoprotein-particle reaction; pancreatic lipase inhibition by orlistat reduces this flux.

Showing all 1 reactions.

What accelerates and inhibits it

Regulation is pathway-specific, so each context is listed separately

0 entries

No regulation recorded for this enzyme in the source documents.

Recent literature

No articles returned.